Controlled Substances Act
Schedule I [21 CFR 1308.11]
Source: Shulgin, Alexander T. Controlled Substances: Chemical & Legal Guide to Federal Drugs Laws (2nd edition). Ronin Publishing Inc., Berkeley, 1992
Source: DEA Office of Diversion Control: Section 1308: Schedules of Controlled Substances
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(g)
Cannabimimetic Agents. Unless specifically exempted or unless listed in another schedule, any material, compound, mixture, or preparation which contains any quantity of cannabimimetic agents, or which contains their salts, isomers, and salts of isomers whenever the existence of such salts, isomers, and salts of isomers is possible within the specific chemical designation.
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(A)
The term ‘cannabimimetic agents’ means any substance that is a cannabinoid receptor type 1 (CB1 receptor) agonist as demonstrated by binding studies and functional assays within any of the following structural classes:
3D rendering of 2-(3-Hydroxycyclohexyl)phenol
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(i)
2-(3-Hydroxycyclohexyl)phenol with substitution at the 5-position of the phenolic ring by alkyl or alkenyl, whether or not substituted on the cyclohexyl ring to any extent.
UK: MDA Part II Class B Section 1(c) 2-(3-Hydroxycyclohexyl)phenol
3D rendering of 3-(1-Naphthoyl)indole
3-(1-Naphthoyl)indole
3D rendering of 3-(1-Naphthylmethane)indole
3-(1-Naphthylmethane)indole
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(ii)
3-(1-Naphthoyl)indole or 3-(1-Naphthylmethane)indole by substitution at the nitrogen atom of the indole ring, whether or not further substituted on the indole ring to any extent, whether or not substituted on the naphthoyl or naphthyl ring to any extent.
CA: CDSA Schedule II Section 2 Subsection 2 3-(1-Naphthoyl)indole
UK: MDA Part II Class B Section 1(c) 3-(1-Naphthoyl)indole
⇒
PubChem: 10355825; ChemSpider: 8531277
UK: MDA Part II Class B Section 1(c) 1H-Indol-3-yl-(1-naphthyl)methane
3D rendering of 3-(1-Naphthoyl)pyrrole
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(iii)
3-(1-Naphthoyl)pyrrole by substitution at the nitrogen atom of the pyrrole ring, whether or not further substituted in the pyrrole ring to any extent, whether or not substituted on the naphthoyl ring to any extent.
CA: CDSA Schedule II Section 2 Subsection 3 3-(1-Naphthoyl)pyrrole
UK: MDA Part II Class B Section 1(c) 3-(1-Naphthoyl)pyrrole
⇒
PubChem: 15832251; ChemSpider: 10506445
3D rendering of 1-(1-Naphthylmethylene)indene
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(iv)
1-(1-Naphthylmethylene)indene by substitution of the 3-position of the indene ring, whether or not further substituted in the indene ring to any extent, whether or not substituted on the naphthyl ring to any extent.
UK: MDA Part II Class B Section 1(c) 1-(1-Naphthylmethylene)indene
3D rendering of 3-Phenylacetylindole
3-Phenylacetylindole
3D rendering of 3-Benzoylindole
3-Benzoylindole
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(v)
3-Phenylacetylindole or 3-Benzoylindole by substitution at the nitrogen atom of the indole ring, whether or not further substituted in the indole ring to any extent, whether or not substituted on the phenyl ring to any extent.
CA: CDSA Schedule II Section 2 Subsection 4 3-Phenylacetylindole
UK: MDA Part II Class B Section 1(c) 3-Phenylacetylindole
⇒
PubChem: 266609; ChemSpider: 234313; Drugs Forum: Phenylacetylindoles
CA: CDSA Schedule II Section 2 Subsection 5 3-Benzoylindole
UK: MDA Part II Class B Section 1(c) 3-Benzoylindole
⇒
PubChem: 84845; ChemSpider: 76537
3D rendering of 5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(1)
7297
5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol (CP 47,497)
CA: CDSA Schedule II Section 2 Subsection 1 5-(1,1-Dimethylheptyl)-2-(3-hydroxycyclohexyl)phenol
UK: MDA Part II Class B Section 1(c) CP 47,497
US: Previously at CSA Schedule I Section h
⇒
PubChem: 15942731; ChemSpider: 10205286; Drugs Forum: CP 47,497; Erowid: Spice Product; Wikipedia: CP 47,497
3D rendering of 5-(1,1-Dimethyloctyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(2)
7298
5-(1,1-Dimethyloctyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol (Cannabicyclohexanol; CP 47,497 C8 homologue)
UK: MDA Part II Class B Section 1(c) CP 47,497-C8
US: Previously at CSA Schedule I Section h
⇒
PubChem: 23986041; Erowid: Spice Product; Wikipedia: Cannabicyclohexanol
3D rendering of 1-Pentyl-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(3)
7118
1-Pentyl-3-(1-naphthoyl)indole (JWH-018; AM678)
CA: CDSA Schedule II Section 2 Subsection 2 1-Pentyl-3-(1-naphthoyl)indole
UK: MDA Part II Class B Section 1(c) JWH-018
US: Previously at CSA Schedule I Section h
⇒
PubChem: 10382701; ChemSpider: 8558143; Bluelight: JWH-018; Drugs Forum: JWH-018; Erowid: Spice Product; Wikipedia: JWH-018
3D rendering of 1-Butyl-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(4)
7173
1-Butyl-3-(1-naphthoyl)indole (JWH-073)
CA: CDSA Schedule II Section 2 Subsection 2 1-Butyl-3-(1-naphthoyl)indole
UK: MDA Part II Class B Section 1(c) JWH-073
US: Previously at CSA Schedule I Section h
⇒
PubChem: 10471670; ChemSpider: 8647081; Bluelight: JWH-073; Erowid: Spice Product; Wikipedia: JWH-073
3D rendering of 1-Hexyl-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(5)
7019
1-Hexyl-3-(1-naphthoyl)indole (JWH-019)
CA: CDSA Schedule II Section 2 Subsection 2 1-Hexyl-3-(1-naphthoyl)indole
⇒
PubChem: 52224389; ChemSpider: 24598813; Wikipedia: JWH-019
3D rendering of 1-[2-(4-Morpholinyl)ethyl]-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(6)
7200
1-[2-(4-Morpholinyl)ethyl]-3-(1-naphthoyl)indole (JWH-200)
CA: CDSA Schedule II Section 2 Subsection 2 1-(2-Morpholin-4-ylethyl)-3-(1naphthoyl)indole
UK: MDA Part II Class B Section 1(c) JWH-200
US: Previously at CSA Schedule I Section h
⇒
PubChem: 10045570; ChemSpider: 8221134; Drugs Forum: JWH-200; Erowid: Spice Product; Wikipedia: JWH-200
3D rendering of 1-Pentyl-3-(2-methoxyphenylacetyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(7)
6250
1-Pentyl-3-(2-methoxyphenylacetyl)indole (JWH-250)
CA: CDSA Schedule II Section 2 Subsection 4 1-Pentyl-3-(2-methoxyphenylacetyl)indole
UK: MDA Part II Class B Section 1(c) JWH-250
⇒
PubChem: 44397540; ChemSpider: 23256117; Drugs Forum: JWH-250; Wikipedia: JWH-250
3D rendering of 1-Pentyl-3-[1-(4-methoxynaphthoyl)]indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(8)
7081
1-Pentyl-3-[1-(4-methoxynaphthoyl)]indole (JWH-081)
CA: CDSA Schedule II Section 2 Subsection 2 1-Butyl-3-(4-methoxy-1-naphthoyl)indole
UK: MDA Part II Class B Section 1(c) JWH-081
⇒
PubChem: 10547208; ChemSpider: 8722599; Wikipedia: JWH-081
3D rendering of 1-Pentyl-3-(4-methyl-1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(9)
7122
1-Pentyl-3-(4-methyl-1-naphthoyl)indole (JWH-122)
CA: CDSA Schedule II Section 2 Subsection 2 1-Pentyl-3-(4-methyl-1-naphthoyl)indole
UK: MDA Part II Class B Section 1(c) JWH-122
⇒
PubChem: 44466638; ChemSpider: 24623066; Bluelight: JWH-122; Wikipedia: JWH-122
3D rendering of 1-Pentyl-3-(4-chloro-1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(10)
7398
1-Pentyl-3-(4-chloro-1-naphthoyl)indole (JWH-398)
UK: MDA Part II Class B Section 1(c) JWH-398
⇒
PubChem: 57458928; ChemSpider: 28647395; Drugs Forum: JWH-398; Wikipedia: JWH-398
3D rendering of 1-(5-Fluoropentyl)-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(11)
7201
1-(5-Fluoropentyl)-3-(1-naphthoyl)indole (AM2201)
CA: CDSA Schedule II Section 2 Subsection 2 1-(5-Fluoropentyl)-3-(1-naphthoyl)indole
UK: MDA Part II Class B Section 1(c) AM-2201
⇒
PubChem: 53393997; ChemSpider: 24751884; Drugs Forum: AM-2201; Wikipedia: AM-2201
3D rendering of 1-(5-Fluoropentyl)-3-(2-iodobenzoyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(12)
7694
1-(5-Fluoropentyl)-3-(2-iodobenzoyl)indole (AM694)
UK: MDA Part II Class B Section 1(c) AM-694
⇒
PubChem: 9889172; ChemSpider: 8064843; Drugs Forum: AM-694; Wikipedia: AM-694
3D rendering of 1-Pentyl-3-[(4-methoxy)-benzoyl]indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(13)
7104
1-Pentyl-3-[(4-methoxy)-benzoyl]indole (SR-19; RCS-4)
UK: MDA Part II Class B Section 1(c) RCS-4 and RCS-4
⇒
PubChem: 56841530; ChemSpider: 24769418; Wikipedia: RCS-4; Wikipedia: RCS-4
3D rendering of 1-Cyclohexylethyl-3-(2-methoxyphenylacetyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(14)
7008
1-Cyclohexylethyl-3-(2-methoxyphenylacetyl)indole (SR-18; RCS-8)
UK: MDA Part II Class B Section 1(c) RCS-8
⇒
PubChem: 53394099; ChemSpider: 24751863; Bluelight: RCS-8; Drugs Forum: RCS-8; Wikipedia: RCS-8
3D rendering of 1-Pentyl-3-(2-chlorophenylacetyl)indole
Effective 4 Jan 2013, 78 FR 664 finalized the prior interim scheduling:
Effective 9 Jul 2012, S. 3187, 112 Cong., 2nd Sess. added:
(15)
7203
1-Pentyl-3-(2-chlorophenylacetyl)indole (JWH-203)
⇒
PubChem: 44397500; ChemSpider: 23256082; Wikipedia: JWH-203
3D rendering of (1-Pentyl-1H-indol-3-yl)(2,2,3,3- tetramethylcyclopropyl)methanone
On 14 May 2015, 80 FR 27611 proposed to add:
(16)
7144
(1-Pentyl-1H-indol-3-yl)(2,2,3,3- tetramethylcyclopropyl)methanone (UR-144)
CA: CDSA Schedule II Section 2 Subsection 6 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- tetramethylcyclopropyl)-methanone
UK: MDA Part II Class B Section 1(c) UR-144
See also CSA Schedule I Section h Subsection 1 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- tetramethylcyclopropyl)methanone
⇒
PubChem: 44626619; ChemSpider: 24634882; Bluelight: UR-144; Drugs Forum: UR-144; Wikipedia: UR-144
3D rendering of [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
On 14 May 2015, 80 FR 27611 proposed to add:
(17)
7011
[1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone (5-Fluoro-UR-144; XLR11)
CA: CDSA Schedule II Section 2 Subsection 6 [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone
UK: MDA Part II Class B Section 1(c) XLR11
See also CSA Schedule I Section h Subsection 2 [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
⇒
PubChem: 57501498; ChemSpider: 28537382; Bluelight: XLR11; Wikipedia: XLR-11 (drug)
3D rendering of N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide
On 14 May 2015, 80 FR 27611 proposed to add:
(18)
7048
N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide (APINACA; AKB48)
CA: CDSA Schedule II Section 2 Subsection 8 N-(Adamantan-1-yl)-1-pentyl-1H-indazole-3-carboxamide
See also CSA Schedule I Section h Subsection 3 N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide
⇒
PubChem: 57404063; ChemSpider: 28189076; Bluelight: AKB48; Drugs Forum: AKB48; Wikipedia: AKB48 (drug)
11 March 2016 · Creative Commons BY-NC-SA ·